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Atomistry » Chlorine » PDB 3k9t-3khf » 3kck | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Atomistry » Chlorine » PDB 3k9t-3khf » 3kck » |
Chlorine in PDB 3kck: A Novel Chemotype of Kinase InhibitorsEnzymatic activity of A Novel Chemotype of Kinase Inhibitors
All present enzymatic activity of A Novel Chemotype of Kinase Inhibitors:
2.7.10.2; Protein crystallography data
The structure of A Novel Chemotype of Kinase Inhibitors, PDB code: 3kck
was solved by
H.J.Zuccola,
T.Wang,
M.W.Ledeboer,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Chlorine Binding Sites:
The binding sites of Chlorine atom in the A Novel Chemotype of Kinase Inhibitors
(pdb code 3kck). This binding sites where shown within
5.0 Angstroms radius around Chlorine atom.
In total only one binding site of Chlorine was determined in the A Novel Chemotype of Kinase Inhibitors, PDB code: 3kck: Chlorine binding site 1 out of 1 in 3kckGo back to Chlorine Binding Sites List in 3kck
Chlorine binding site 1 out
of 1 in the A Novel Chemotype of Kinase Inhibitors
Mono view Stereo pair view
Reference:
T.Wang,
M.W.Ledeboer,
J.P.Duffy,
A.C.Pierce,
H.J.Zuccola,
E.Block,
D.Shlyakter,
J.K.Hogan,
Y.L.Bennani.
A Novel Chemotype of Kinase Inhibitors: Discovery of 3,4-Ring Fused 7-Azaindoles and Deazapurines As Potent JAK2 Inhibitors. Bioorg.Med.Chem.Lett. V. 20 153 2010.
Page generated: Sat Dec 12 09:50:49 2020
ISSN: ISSN 0960-894X PubMed: 19945871 DOI: 10.1016/J.BMCL.2009.11.021 |
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