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Atomistry » Chlorine » PDB 5hi4-5hpu » 5hm0 » |
Chlorine in PDB 5hm0: Crystal Structure of the First Bromodomain of Human BRD4 Bound to Benzoisoxazoloazepine 3Protein crystallography data
The structure of Crystal Structure of the First Bromodomain of Human BRD4 Bound to Benzoisoxazoloazepine 3, PDB code: 5hm0
was solved by
H.Jayaram,
F.Poy,
J.W.Setser,
S.F.Bellon,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Chlorine Binding Sites:
The binding sites of Chlorine atom in the Crystal Structure of the First Bromodomain of Human BRD4 Bound to Benzoisoxazoloazepine 3
(pdb code 5hm0). This binding sites where shown within
5.0 Angstroms radius around Chlorine atom.
In total only one binding site of Chlorine was determined in the Crystal Structure of the First Bromodomain of Human BRD4 Bound to Benzoisoxazoloazepine 3, PDB code: 5hm0: Chlorine binding site 1 out of 1 in 5hm0Go back to Chlorine Binding Sites List in 5hm0
Chlorine binding site 1 out
of 1 in the Crystal Structure of the First Bromodomain of Human BRD4 Bound to Benzoisoxazoloazepine 3
Mono view Stereo pair view
Reference:
B.K.Albrecht,
V.S.Gehling,
M.C.Hewitt,
R.G.Vaswani,
A.Cote,
Y.Leblanc,
C.G.Nasveschuk,
S.Bellon,
L.Bergeron,
R.Campbell,
N.Cantone,
M.R.Cooper,
R.T.Cummings,
H.Jayaram,
S.Joshi,
J.A.Mertz,
A.Neiss,
E.Normant,
M.O'meara,
E.Pardo,
F.Poy,
P.Sandy,
J.Supko,
R.J.Sims,
J.C.Harmange,
A.M.Taylor,
J.E.Audia.
Identification of A Benzoisoxazoloazepine Inhibitor (Cpi-0610) of the Bromodomain and Extra-Terminal (Bet) Family As A Candidate For Human Clinical Trials. J.Med.Chem. V. 59 1330 2016.
Page generated: Sat Dec 12 11:48:53 2020
ISSN: ISSN 0022-2623 PubMed: 26815195 DOI: 10.1021/ACS.JMEDCHEM.5B01882 |
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