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Atomistry » Chlorine » PDB 4tsz-4u2x » 4tvk | ||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Atomistry » Chlorine » PDB 4tsz-4u2x » 4tvk » |
Chlorine in PDB 4tvk: Torpedo Californica Acetylcholinesterase in Complex with A Chlorotacrine-Juglone Hybrid InhibitorEnzymatic activity of Torpedo Californica Acetylcholinesterase in Complex with A Chlorotacrine-Juglone Hybrid Inhibitor
All present enzymatic activity of Torpedo Californica Acetylcholinesterase in Complex with A Chlorotacrine-Juglone Hybrid Inhibitor:
3.1.1.7; Protein crystallography data
The structure of Torpedo Californica Acetylcholinesterase in Complex with A Chlorotacrine-Juglone Hybrid Inhibitor, PDB code: 4tvk
was solved by
A.Pesaresi,
S.Samez,
D.Lamba,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Chlorine Binding Sites:
The binding sites of Chlorine atom in the Torpedo Californica Acetylcholinesterase in Complex with A Chlorotacrine-Juglone Hybrid Inhibitor
(pdb code 4tvk). This binding sites where shown within
5.0 Angstroms radius around Chlorine atom.
In total only one binding site of Chlorine was determined in the Torpedo Californica Acetylcholinesterase in Complex with A Chlorotacrine-Juglone Hybrid Inhibitor, PDB code: 4tvk: Chlorine binding site 1 out of 1 in 4tvkGo back to![]() ![]()
Chlorine binding site 1 out
of 1 in the Torpedo Californica Acetylcholinesterase in Complex with A Chlorotacrine-Juglone Hybrid Inhibitor
![]() Mono view ![]() Stereo pair view
Reference:
E.Nepovimova,
E.Uliassi,
J.Korabecny,
L.E.Pena-Altamira,
S.Samez,
A.Pesaresi,
G.E.Garcia,
M.Bartolini,
V.Andrisano,
C.Bergamini,
R.Fato,
D.Lamba,
M.Roberti,
K.Kuca,
B.Monti,
M.L.Bolognesi.
Multitarget Drug Design Strategy: Quinone-Tacrine Hybrids Designed to Block Amyloid-Beta Aggregation and to Exert Anticholinesterase and Antioxidant Effects. J.Med.Chem. V. 57 8576 2014.
Page generated: Fri Jul 26 01:56:08 2024
ISSN: ISSN 0022-2623 PubMed: 25259726 DOI: 10.1021/JM5010804 |
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