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Chlorine in PDB 6t2k: Furano[2,3-D]Prymidine Amides As Notum InhibitorsEnzymatic activity of Furano[2,3-D]Prymidine Amides As Notum Inhibitors
All present enzymatic activity of Furano[2,3-D]Prymidine Amides As Notum Inhibitors:
3.1.1.98; Protein crystallography data
The structure of Furano[2,3-D]Prymidine Amides As Notum Inhibitors, PDB code: 6t2k
was solved by
Y.Zhao,
E.Y.Jones,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Chlorine Binding Sites:
The binding sites of Chlorine atom in the Furano[2,3-D]Prymidine Amides As Notum Inhibitors
(pdb code 6t2k). This binding sites where shown within
5.0 Angstroms radius around Chlorine atom.
In total only one binding site of Chlorine was determined in the Furano[2,3-D]Prymidine Amides As Notum Inhibitors, PDB code: 6t2k: Chlorine binding site 1 out of 1 in 6t2kGo back to Chlorine Binding Sites List in 6t2k
Chlorine binding site 1 out
of 1 in the Furano[2,3-D]Prymidine Amides As Notum Inhibitors
Mono view Stereo pair view
Reference:
B.N.Atkinson,
D.Steadman,
W.Mahy,
Y.Zhao,
J.Sipthorp,
E.D.Bayle,
F.Svensson,
G.Papageorgiou,
F.Jeganathan,
S.Frew,
A.Monaghan,
M.Bictash,
E.Y.Jones,
P.V.Fish.
Scaffold-Hopping Identifies Furano[2,3-D]Pyrimidine Amides As Potent Notum Inhibitors. Bioorg.Med.Chem.Lett. 26751 2019.
Page generated: Sat Dec 12 13:41:58 2020
ISSN: ESSN 1464-3405 PubMed: 31862412 DOI: 10.1016/J.BMCL.2019.126751 |
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